Wednesday, February 21, 2018

PIRENZIPINE SUBTYPYPE OF MUSCARINIC RECEPTOR ANTAGONIST ITS USES AND SIDE EFFECTS

MECHANISM OF ACTION- 
It is a muscarinic receptor antagonist and binds to the muscarinic acetylcholine receptor. The Muscarinic acetylcholine receptor mediates various cellular responses, including inhibition of adenylate cyclase, breakdown of phosphoinositides and modulation of potassium channels through the action of G protein.

USES-
1. Antisecretory action
2. Peptic ulcer
3. Antispasmodic
4. Bronchial asthama
5. Mydriatic

SIDE EFFECTS-
1. Dry mouth
2. Rashes
3. Fever
4. Photophobia
5. Blurred vision

PHARMACOLOGICAL  ACTION-
It stimulates medullary centre.
It produces tachycardia.
Visceral smooth muscles are relaxed.
Decreases sweat , salivary or tracheobronchial secretion.

DRUG-DRUG INTERACTION- 
Cimetidine + Pirenzipine = lowers gastric secretion.

REFERENCE 


Tripathi K.D,"Essentials of medical pharmacology",7th edition,page no.101

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