Sunday, March 18, 2018

Diethylstilbesterol


MECHANISM OF ACTION-
1. Estrogens diffuse into the target cells and binds with a protein receptor, known as estrogen receptor, which are present in the female reproductive tract, the mammary gland, the hypothalamus, and the pituitary.
2. The  binding of estrogen to the receptors leads to the formation of estrogen receptor complex, which results in the increase of hepatic synthesis of sex hormone binding globulin (SHBG), thyroid-binding globulin (TBG), and other serum proteins and also suppress follicle-stimulating hormone (FSH) from the anterior pituitary.
3. Estrogen along with progestin suppresses the hypothalamic-pituitary system, hence decreasing the secretion of gonadotropin-releasing hormone (GnRH).



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