Sunday, March 18, 2018

Mesna



MECHANISM OF ACTION-

  1. Acrolein (metabolite) is produced when ifosfamide and cyclophosphamide are metabolized.  
  2. This metabolite concentrates in the bladder and causes cell death through upregulation of reactive oxygen species (ROS), and  also activates inducible nitric oxide synthase (iNOS) which leads to the production of nitric oxide (NO).
  3.  Both ROS and NO produce products which are harmful to lipids, proteins and DNA strands.



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